Direct alkylation of heteroaryls using potassium alkyl- and alkoxymethyltrifluoroborates.

ABSTRACT: A direct alkylation of various heteroaryls using stoichiometric potassium alkyl- and alkoxymethyltrifluoroborates has been developed. This method leads to the synthesis of complex substituted heterocycles, which have been obtained with yields up to 89%.

SUBMITTER: Molander GA 

PROVIDER: S-EPMC3069859 | biostudies-literature | 2011 Apr

REPOSITORIES: biostudies-literature