A Protocol for Direct Stereospecific Amination of Primary, Secondary, and Tertiary Alkylboronic Esters.

ABSTRACT: The direct, stereospecific amination of alkylboronic and borinic esters can be conducted by treatment of the organoboron compound with methoxyamine and potassium tert-butoxide. In addition to being stereospecific, this process also enables the direct amination of tertiary boronic esters in an efficient fashion.

SUBMITTER: Edelstein EK 

PROVIDER: S-EPMC6322687 | biostudies-literature | 2018 Aug

REPOSITORIES: biostudies-literature